- Molecular NameOmeprazole
- SynonymOMEP; Omeprazol [INN-Spanish]; omeprazole; Omeprazole magnesium; Omeprazolum [INN-Latin]; OMP; OMZ
- Weight345.423
- Drugbank_IDDB00338
- ACS_NO73590-58-6
- Show 3D model
- LogP (experiment)2.23
- LogP (predicted, AB/LogP v2.0)2.44
- pka4.0
- LogD (pH=7, predicted)2.43
- Solubility (experiment)0.131 mg/ml
- LogS (predicted, ACD/Labs)(ph=7)-3.95
- LogSw (predicted, AB/LogsW2.0)0.26
- Sw (mg/ml) (predicted, ACD/Labs)0.04
- No.of HBond Donors1
- No.of HBond Acceptors6
- No.of Rotatable Bonds5
- TPSA96.31
- StatusFDA approved
- AdministrationOral, IV
- PharmacologyA proton pump inhibitor used in the treatment of dyspepsia, peptic ulcer disease (PUD), gastroesophageal reflux disease (GORD/GERD) and Zollinger-Ellison syndrome.
- Absorption_value80.0
- Absorption (description)N/A
- Caco_2N/A
- Bioavailability47.0
- Protein binding95.0
- Volume of distribution (VD)0.27 to 0.45 L/kg
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmHepatic (CYP2C19, CYP3A4)
- Half life0.5~3 h
- Excretion80% Renal, 20% Faecal
- Urinary ExcretionN/A
- CleranceN/A
- ToxicitySymptoms of overdose include confusion, drowsiness, blurred vision, tachycardia, nausea, diaphoresis, flushing, headache, and dry mouth.
- LD50 (rat)N/A
- LD50 (mouse)N/A