- Molecular NamePenicillin_G
- SynonymNA
- Weight333.388
- Drugbank_IDDB01053
- ACS_NO61-33-6
- Show 3D model
- LogP (experiment)1.83
- LogP (predicted, AB/LogP v2.0)2.08
- pka2.8
- LogD (pH=7, predicted)-1.88
- Solubility (experiment)0.21 mg/ml
- LogS (predicted, ACD/Labs)(ph=7)0.48
- LogSw (predicted, AB/LogsW2.0)1.02
- Sw (mg/ml) (predicted, ACD/Labs)0.82
- No.of HBond Donors2
- No.of HBond Acceptors6
- No.of Rotatable Bonds4
- TPSA112.01
- StatusFDA approved
- Administrationintravenous bolus
- PharmacologyPenicillin G is a penicillin beta-lactam antibiotic used in the treatment of bacterial infections caused by susceptible, usually gram-positive, organisms.
- Absorption_valueN/A
- Absorption (description)Rapidly absorbed following both intramuscular and subcutaneous injection. Initial blood levels following parenteral administration are high but transient.
- Caco_2N/A
- BioavailabilityN/A
- Protein binding60.0
- Volume of distribution (VD)0.6 L/kg
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmHepatic
- Half life0.5 h
- Excretionrenal
- Urinary Excretion79
- Clerance5~9 ml/min/kg
- ToxicityNeurological adverse reactions, including convulsions, may occur with the attainment of high CSF levels of beta-lactams.
- LD50 (rat)8900 mk/kg
- LD50 (mouse)N/A