- Molecular NameZanamivir
- SynonymGANA; GNA; Modified sialic acid; Zanamavir; ZMR
- Weight332.313
- Drugbank_IDDB00558
- ACS_NO139110-80-8
- Show 2D model
- LogP (experiment)N/A
- LogP (predicted, AB/LogP v2.0)-3.31
- pkaN/A
- LogD (pH=7, predicted)-5.81
- Solubility (experiment)N/A
- LogS (predicted, ACD/Labs)(ph=7)-0.43
- LogSw (predicted, AB/LogsW2.0)34.33
- Sw (mg/ml) (predicted, ACD/Labs)123.97
- No.of HBond Donors9
- No.of HBond Acceptors11
- No.of Rotatable Bonds7
- TPSA198.22
- StatusFDA approved
- AdministrationInhalation
- PharmacologyA neuraminidase inhibitor used in the treatment and prophylaxis of Influenzavirus A and Influenzavirus B.
- Absorption_value2.0
- Absorption (description)N/A
- Caco_2N/A
- Bioavailability2.0
- Protein binding10.0
- Volume of distribution (VD)16 L; decreases in patients with renal impairment (13.4 L in those with severe impairment; 15.1 L for mild–moderate impairment).
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmNot metabolized
- Half life2.5~5.1 h
- ExcretionRenal
- Urinary ExcretionN/A
- CleranceN/A
- ToxicityN/A
- LD50 (rat)N/A
- LD50 (mouse)N/A