- Molecular NameQuinidine
- SynonymQuinidine Gluconate; Quinidine Sulfate
- Weight324.424
- Drugbank_IDDB00908
- ACS_NO56-54-2
- Show 2D model
- LogP (experiment)2.64
- LogP (predicted, AB/LogP v2.0)2.89
- pka4.2, 8.8
- LogD (pH=7, predicted)1.32
- Solubility (experiment)0.142 mg/ml
- LogS (predicted, ACD/Labs)(ph=7)-1.2
- LogSw (predicted, AB/LogsW2.0)0.28
- Sw (mg/ml) (predicted, ACD/Labs)0.15
- No.of HBond Donors1
- No.of HBond Acceptors4
- No.of Rotatable Bonds4
- TPSA45.59
- StatusFDA approved
- AdministrationN/A
- PharmacologyA pharmaceutical agent that acts as a class I antiarrhythmic agent (Ia) in the heart. It is a stereoisomer of quinine, originally derived from the bark of the cinchona tree.
- Absorption_value80.0
- Absorption (description)N/A
- Caco_2-4.69
- Bioavailability75.0
- Protein binding87.0
- Volume of distribution (VD)3.5 L/kg
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmMetabolically cleared primarily by CYP3A
- Half life6.2 h
- ExcretionRenal
- Urinary Excretion18
- Clerance4.7 ml/min/kg
- ToxicityN/A
- LD50 (rat)N/A
- LD50 (mouse)LD50=594