- Molecular NameButenafine
- SynonymButenafina [INN-Spanish]; Butenafine [INN]; Butenafine HCL; Butenafine hydrochloride; Butenafinum [INN-Latin]…
- Weight317.476
- Drugbank_IDDB01091
- ACS_NO101828-21-1
- Show 2D model
- LogP (experiment)7.12
- LogP (predicted, AB/LogP v2.0)6.2
- pkaN/A
- LogD (pH=7, predicted)5.72
- Solubility (experiment)N/A
- LogS (predicted, ACD/Labs)(ph=7)-4.66
- LogSw (predicted, AB/LogsW2.0)0.0
- Sw (mg/ml) (predicted, ACD/Labs)0.0
- No.of HBond Donors0
- No.of HBond Acceptors1
- No.of Rotatable Bonds5
- TPSA3.24
- StatusFDA approved
- Administrationtopical
- PharmacologyA synthetic benzylamine antifungal, marketed under the trade names Mentax, Butop (India) and is the active ingredient in Schering-Plough's Lotrimin Ultra.
- Absorption_valueN/A
- Absorption (description)N/A
- Caco_2N/A
- BioavailabilityN/A
- Protein bindingN/A
- Volume of distribution (VD)N/A
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmHeptatic. The primary metabolite in urine was formed through hydroxylation at the terminal t-butyl side-chain.
- Half life35~100 h
- ExcretionN/A
- Urinary ExcretionN/A
- CleranceN/A
- ToxicityN/A
- LD50 (rat)N/A
- LD50 (mouse)N/A