- Molecular NameMinaprine
- SynonymMinaprina [INN-Spanish]; Minaprine Dihydrochloride; Minaprine Hydrochloride; Minaprinum [INN-Latin]
- Weight298.39
- Drugbank_IDDB00805
- ACS_NO25905-77-5
- Show 2D model
- LogP (experiment)2.03
- LogP (predicted, AB/LogP v2.0)2.23
- pkaN/A
- LogD (pH=7, predicted)2.01
- Solubility (experiment)2.36 mg/ml
- LogS (predicted, ACD/Labs)(ph=7)-1.61
- LogSw (predicted, AB/LogsW2.0)0.78
- Sw (mg/ml) (predicted, ACD/Labs)4.09
- No.of HBond Donors1
- No.of HBond Acceptors5
- No.of Rotatable Bonds5
- TPSA50.28
- StatusFDA approved; US withdrawn
- AdministrationN/A
- PharmacologyAn antidepressant drug which acts as a weak, short-acting monoamine oxidase inhibitor, acting mainly at the MAOA subtype.
- Absorption_valueN/A
- Absorption (description)N/A
- Caco_2N/A
- BioavailabilityN/A
- Protein bindingN/A
- Volume of distribution (VD)N/A
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmHepatic. Cytochrome P4502D is responsible for the 4-hydroxylation of minaprine to 4-hydroxyminaprine.
- Half lifeN/A
- ExcretionN/A
- Urinary ExcretionN/A
- CleranceN/A
- ToxicityN/A
- LD50 (rat)N/A
- LD50 (mouse)LD50=37 (intraperitoneal)