- Molecular NamePenbutolol
- SynonymPenbutolol sulfate
- Weight291.435
- Drugbank_IDDB01359
- ACS_NO36507-48-9
- Show 3D model
- LogP (experiment)4.15
- LogP (predicted, AB/LogP v2.0)3.89
- pkaN/A
- LogD (pH=7, predicted)1.41
- Solubility (experiment)N/A
- LogS (predicted, ACD/Labs)(ph=7)-0.68
- LogSw (predicted, AB/LogsW2.0)2.06
- Sw (mg/ml) (predicted, ACD/Labs)0.25
- No.of HBond Donors2
- No.of HBond Acceptors3
- No.of Rotatable Bonds7
- TPSA41.49
- StatusFDA approved
- AdministrationN/A
- PharmacologyA medication in the class of beta blockers, used in the treatment of high blood pressure.
- Absorption_value100.0
- Absorption (description)N/A
- Caco_2N/A
- Bioavailability90.0
- Protein binding89.0
- Volume of distribution (VD)5.1 L/kg
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmPenbutolol is extensively metabolized in the liver by hydroxylation and glucuronidation. Active metabolites have not been identified
- Half lifeN/A
- ExcretionN/A
- Urinary ExcretionN/A
- CleranceN/A
- ToxicityN/A
- LD50 (rat)N/A
- LD50 (mouse)N/A