- Molecular NameQuinethazone
- SynonymChinetazone [dcit]; Chinethazonum; Quinetazona [inn-spanish]; Quinethazon; Quinethazonum [inn-latin]
- Weight289.743
- Drugbank_IDDB01325
- ACS_NO73-49-4
- Show 2D model
- LogP (experiment)0.2
- LogP (predicted, AB/LogP v2.0)1.05
- pka9.3, 10.7
- LogD (pH=7, predicted)1.04
- Solubility (experiment)0.149 mg/ml
- LogS (predicted, ACD/Labs)(ph=7)-3.15
- LogSw (predicted, AB/LogsW2.0)0.32
- Sw (mg/ml) (predicted, ACD/Labs)0.2
- No.of HBond Donors4
- No.of HBond Acceptors6
- No.of Rotatable Bonds2
- TPSA109.67
- StatusFDA approved
- AdministrationN/A
- PharmacologyA thiazide diuretic used to treat hypertension. Common side effects include dizziness, dry mouth, nausea, and low potassium levels.
- Absorption_valueN/A
- Absorption (description)N/A
- Caco_2N/A
- BioavailabilityN/A
- Protein bindingN/A
- Volume of distribution (VD)N/A
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmN/A
- Half lifeN/A
- ExcretionN/A
- Urinary ExcretionN/A
- CleranceN/A
- ToxicityN/A
- LD50 (rat)N/A
- LD50 (mouse)N/A