- Molecular NameDyclonine
- SynonymNA
- Weight289.419
- Drugbank_IDDB00645
- ACS_NO586-60-7
- Show 2D model
- LogP (experiment)3.931
- LogP (predicted, AB/LogP v2.0)4.03
- pkaN/A
- LogD (pH=7, predicted)2.09
- Solubility (experiment)N/A
- LogS (predicted, ACD/Labs)(ph=7)-2.08
- LogSw (predicted, AB/LogsW2.0)0.24
- Sw (mg/ml) (predicted, ACD/Labs)0.06
- No.of HBond Donors0
- No.of HBond Acceptors3
- No.of Rotatable Bonds8
- TPSA29.54
- StatusFDA approved
- AdministrationN/A
- PharmacologyAn oral anaesthetic found in Sucrets, an over the counter throat lozenge. It is also found in some varieties of the Cepacol sore throat spray.
- Absorption_valueN/A
- Absorption (description)N/A
- Caco_2N/A
- BioavailabilityN/A
- Protein bindingN/A
- Volume of distribution (VD)N/A
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmN/A
- Half life30~60 min
- ExcretionN/A
- Urinary ExcretionN/A
- CleranceN/A
- ToxicitySymptoms of overdose include cardiovascular system depression, CNS toxicity, and methemoglobinemia.
- LD50 (rat)N/A
- LD50 (mouse)LD50=130 (intraperitoneal)