- Molecular NameLenalidomide
- SynonymCC-5013; CDC 501; IMiD3; lenalidomide
- Weight259.265
- Drugbank_IDDB00480
- ACS_NO191732-72-6
- Show 2D model
- LogP (experiment)-0.318
- LogP (predicted, AB/LogP v2.0)0.43
- pkaN/A
- LogD (pH=7, predicted)0.41
- Solubility (experiment)N/A
- LogS (predicted, ACD/Labs)(ph=7)-1.13
- LogSw (predicted, AB/LogsW2.0)1.14
- Sw (mg/ml) (predicted, ACD/Labs)19.32
- No.of HBond Donors3
- No.of HBond Acceptors6
- No.of Rotatable Bonds1
- TPSA92.5
- StatusFDA approved
- AdministrationN/A
- PharmacologyA treatment for multiple myeloma, for which thalidomide is an accepted therapeutic modality, but has also shown efficacy in the class of hematological disorders known as myelodysplastic syndromes (MDS).
- Absorption_valueN/A
- Absorption (description)N/A
- Caco_2N/A
- BioavailabilityN/A
- Protein binding30.0
- Volume of distribution (VD)N/A
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmUndetermined
- Half life3 h
- ExcretionRenal (67% unchanged)
- Urinary ExcretionN/A
- CleranceN/A
- ToxicityThe most frequently reported adverse events were related to blood and lymphatic system disorders, skin and subcutaneous tissue disorders, gastrointestinal disorders, and general disorders and administrative site conditions.
- LD50 (rat)N/A
- LD50 (mouse)N/A