- Molecular NameEthoxzolamide
- SynonymEthoxazolamide; Ethoxyzolamide; Etoxzolamide
- Weight258.322
- Drugbank_IDDB00311
- ACS_NO452-35-7
- Show 2D model
- LogP (experiment)2.01
- LogP (predicted, AB/LogP v2.0)1.88
- pka8.1
- LogD (pH=7, predicted)1.85
- Solubility (experiment)0.0241 mg/ml
- LogS (predicted, ACD/Labs)(ph=7)-3.47
- LogSw (predicted, AB/LogsW2.0)0.09
- Sw (mg/ml) (predicted, ACD/Labs)0.09
- No.of HBond Donors2
- No.of HBond Acceptors5
- No.of Rotatable Bonds3
- TPSA118.9
- StatusFDA approved
- AdministrationN/A
- PharmacologyA sulfonamide medication that functions as a carbonic anhydrase inhibitor. It is used in the treatment of glaucoma, duodenal ulcers, and as a diuretic. It may also be used in the treatment of some forms of epilepsy.
- Absorption_valueN/A
- Absorption (description)N/A
- Caco_2N/A
- Bioavailability65.0
- Protein binding89.0
- Volume of distribution (VD)N/A
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmN/A
- Half life2.5~5.5 h
- ExcretionN/A
- Urinary ExcretionN/A
- CleranceN/A
- ToxicityN/A
- LD50 (rat)N/A
- LD50 (mouse)N/A