- Molecular NameMethyldopate
- SynonymAlpha medopa; Alphamethyldopa; AMD; L-Methyl Dopa; Methyldopa anhydrous; Methyldopate; Methyldopate HCL; Mk; B51
- Weight239.271
- Drugbank_IDN/A
- ACS_NO113-42-8
- Show 3D model
- LogP (experiment)N/A
- LogP (predicted, AB/LogP v2.0)0.6
- pkaN/A
- LogD (pH=7, predicted)-0.27
- Solubility (experiment)N/A
- LogS (predicted, ACD/Labs)(ph=7)-0.58
- LogSw (predicted, AB/LogsW2.0)11.84
- Sw (mg/ml) (predicted, ACD/Labs)23.95
- No.of HBond Donors4
- No.of HBond Acceptors5
- No.of Rotatable Bonds5
- TPSA92.78
- StatusN/A
- AdministrationN/A
- PharmacologyA synthetic analogue of ergonovine, a psychedelic alkaloid found in ergot, and many species of morning glory. It is a member of the ergoline family and chemically similar to LSD, ergine, ergometrine, and lysergic acid. Due to its oxytocic properties, it has a medical use in obstetrics.
- Absorption_valueN/A
- Absorption (description)N/A
- Caco_2N/A
- BioavailabilityN/A
- Protein bindingN/A
- Volume of distribution (VD)2 L/kg
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmN/A
- Half life4 h
- ExcretionN/A
- Urinary ExcretionN/A
- CleranceN/A
- ToxicityN/A
- LD50 (rat)N/A
- LD50 (mouse)N/A