- Molecular NameNabumetone
- SynonymNabumetona; Nabumetonum [INN-Latin]
- Weight228.291
- Drugbank_IDDB00461
- ACS_NO42924-53-8
- Show 3D model
- LogP (experiment)3.08
- LogP (predicted, AB/LogP v2.0)3.44
- pkaN/A
- LogD (pH=7, predicted)3.44
- Solubility (experiment)0.0587 mg/ml
- LogS (predicted, ACD/Labs)(ph=7)-3.42
- LogSw (predicted, AB/LogsW2.0)0.03
- Sw (mg/ml) (predicted, ACD/Labs)0.09
- No.of HBond Donors0
- No.of HBond Acceptors2
- No.of Rotatable Bonds4
- TPSA26.3
- StatusFDA approved
- AdministrationN/A
- PharmacologyA non-steroidal anti-inflammatory drug
- Absorption_value80.0
- Absorption (description)N/A
- Caco_2N/A
- Bioavailability35.0
- Protein bindingN/A
- Volume of distribution (VD)7.5 L (steady state); ranges between 5 and 10 L (0.1 to 0.2 L/kg).
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmHepatic, to active metabolite 6-methoxy-2-naphthylacetic acid; 6-MNA
- Half life6-MNA, 22 to 27 h (young healthy subjects), 25 to 34 h (elderly).
- ExcretionRenal
- Urinary ExcretionN/A
- CleranceN/A
- ToxicityN/A
- LD50 (rat)N/A
- LD50 (mouse)N/A