- Molecular NameSulfacetamide
- SynonymNA
- Weight214.245
- Drugbank_IDDB00634
- ACS_NO144-80-9
- Show 3D model
- LogP (experiment)-1.0
- LogP (predicted, AB/LogP v2.0)-0.52
- pka1.8, 5.4
- LogD (pH=7, predicted)-2.24
- Solubility (experiment)6.62 mg/ml
- LogS (predicted, ACD/Labs)(ph=7)0.12
- LogSw (predicted, AB/LogsW2.0)6.77
- Sw (mg/ml) (predicted, ACD/Labs)15.19
- No.of HBond Donors3
- No.of HBond Acceptors5
- No.of Rotatable Bonds2
- TPSA97.64
- StatusFDA approved
- AdministrationN/A
- PharmacologyA sulfonamide antibiotic.
- Absorption_valueN/A
- Absorption (description)N/A
- Caco_2N/A
- BioavailabilityN/A
- Protein binding82.5
- Volume of distribution (VD)N/A
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmN/A
- Half life2.5 h
- ExcretionN/A
- Urinary ExcretionN/A
- CleranceN/A
- ToxicitySide effects include moderate to severe erythema (redness) and moderate edema (raised kin), nausea, vomiting, headache, dizziness, and tiredness. Higher exposure causes unconsciousness.
- LD50 (rat)N/A
- LD50 (mouse)LD50=16500 mg/kg