- Molecular NameThiabendazole
- SynonymTBDZ; TBZ; Thiabendazol; Thiabendole; Thiabenzazole; Thiabenzole; Tiabendazol; Tiabendazole
- Weight201.253
- Drugbank_IDDB00730
- ACS_NO148-79-8
- Show 2D model
- LogP (experiment)2.47
- LogP (predicted, AB/LogP v2.0)2.42
- pka4.64
- LogD (pH=7, predicted)2.42
- Solubility (experiment)0.028 mg/ml
- LogS (predicted, ACD/Labs)(ph=7)-3.53
- LogSw (predicted, AB/LogsW2.0)0.1
- Sw (mg/ml) (predicted, ACD/Labs)0.06
- No.of HBond Donors1
- No.of HBond Acceptors3
- No.of Rotatable Bonds1
- TPSA69.81
- StatusFDA approved
- AdministrationN/A
- PharmacologyA fungicide and parasiticide.
- Absorption_value90.0
- Absorption (description)Rapidly absorbed and peak plasma concentration is reached within 1 to 2 hours after the oral administration of a suspension. Some systemic absorption may occur from topical preparations applied to the skin.
- Caco_2N/A
- BioavailabilityN/A
- Protein bindingN/A
- Volume of distribution (VD)N/A
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmHepatic. Metabolized almost completely to the 5-hydroxy form which appears in the urine as glucuronide or sulfate conjugates.
- Half life8 h
- Excretion90% Urine; 5% Faeces
- Urinary ExcretionN/A
- CleranceN/A
- ToxicityOverdosage may be associated with transient disturbances of vision and psychic alterations.
- LD50 (rat)LD50=3.1 g/kg
- LD50 (mouse)LD50=3.6 g/kg