- Molecular NameAminohippurate
- SynonymAminohippurate Sodium; Aminohippuric acid; Aminohippuric acid Sodium salt; PAH; para-Aminohippurate; Sodium p-aminohippurate; Sodium para-Aminohippurate
- Weight194.19
- Drugbank_IDDB00345
- ACS_NO61-78-9
- Show 3D model
- LogP (experiment)-0.052
- LogP (predicted, AB/LogP v2.0)-0.89
- pka3.6
- LogD (pH=7, predicted)-4.31
- Solubility (experiment)Slightly soluble
- LogS (predicted, ACD/Labs)(ph=7)0.71
- LogSw (predicted, AB/LogsW2.0)19.76
- Sw (mg/ml) (predicted, ACD/Labs)32.06
- No.of HBond Donors4
- No.of HBond Acceptors5
- No.of Rotatable Bonds3
- TPSA92.42
- StatusFDA approved
- AdministrationN/A
- PharmacologyA diagnostic agent useful in medical tests involving the kidney used in the measurement of renal plasma flow.
- Absorption_valueN/A
- Absorption (description)N/A
- Caco_2N/A
- BioavailabilityN/A
- Protein bindingN/A
- Volume of distribution (VD)N/A
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmN/A
- Half life0.2 h
- ExcretionAminohippuric acid is a major metabolite of aminobenzoic acid. After intravenous administration it is rapidly excreted in the urine in subjects with normal renal function.
- Urinary ExcretionN/A
- CleranceN/A
- ToxicityThe intravenous LD50 in female mice is 7.22 g/kg.
- LD50 (rat)N/A
- LD50 (mouse)N/A