- Molecular NamePropofol
- Synonym2,6-Diisopropylphenol; Diisopropylphenol
- Weight178.275
- Drugbank_IDDB00818
- ACS_NO2078-54-8
- Show 3D model
- LogP (experiment)3.79
- LogP (predicted, AB/LogP v2.0)3.74
- pka11.1
- LogD (pH=7, predicted)3.74
- Solubility (experiment)0.124 mg/ml
- LogS (predicted, ACD/Labs)(ph=7)-3.03
- LogSw (predicted, AB/LogsW2.0)0.01
- Sw (mg/ml) (predicted, ACD/Labs)0.17
- No.of HBond Donors1
- No.of HBond Acceptors1
- No.of Rotatable Bonds2
- TPSA20.23
- StatusFDA approved
- AdministrationIntravenous
- PharmacologyA short-acting, intravenously administered hypnotic agent. Its uses include the induction and maintenance of general anesthesia, sedation for mechanically ventilated adults, and procedural sedation. Propofol is also commonly used in veterinary medicine.
- Absorption_value100.0
- Absorption (description)N/A
- Caco_2N/A
- BioavailabilityN/A
- Protein binding98.5
- Volume of distribution (VD)1.7 L/kg
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmPropofol is extensively metabolized by UGTs.
- Half life3.5 h
- ExcretionN/A
- Urinary ExcretionN/A
- Clerance27 ml/min/kg
- ToxicityN/A
- LD50 (rat)N/A
- LD50 (mouse)LD50=32