- Molecular NamePaclitaxel
- Synonym7-epi-Paclitaxel; 7-epi-Taxol; 7-Epipaclitaxel; 7-Epitaxol; ABI-007
- Weight853.918
- Drugbank_IDDB01229
- ACS_NO33069-62-4
- Show 3D model
- LogP (experiment)N/A
- LogP (predicted, AB/LogP v2.0)3.28
- pkaN/A
- LogD (pH=7, predicted)3.28
- Solubility (experiment)N/A
- LogS (predicted, ACD/Labs)(ph=7)-7.25
- LogSw (predicted, AB/LogsW2.0)0.0
- Sw (mg/ml) (predicted, ACD/Labs)0.0
- No.of HBond Donors4
- No.of HBond Acceptors15
- No.of Rotatable Bonds14
- TPSA221.29
- StatusFDA approved
- AdministrationIV
- PharmacologyA mitotic inhibitor used in cancer chemotherapy.
- Absorption_valueN/A
- Absorption (description)N/A
- Caco_2N/A
- Bioavailability6.5
- Protein binding93.0
- Volume of distribution (VD)2.4 L/kg
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmMetabolized by CYP2C8 and CYP3A, and substrate for P-glycoprotein.
- Half life3 h (Average accumulation t1/2; longer terminal t?? s up to 30 hours are reported)
- ExcretionFecal and urinary
- Urinary Excretion5
- Clerance5.5 ml/min/kg
- ToxicityN/A
- LD50 (rat)N/A
- LD50 (mouse)N/A