- Molecular NameAcetyldigitoxin
- SynonymNA
- Weight806.987
- Drugbank_IDDB00511
- ACS_NO1111-393
- Show 3D model
- LogP (experiment)3.779
- LogP (predicted, AB/LogP v2.0)3.01
- pkaN/A
- LogD (pH=7, predicted)3.01
- Solubility (experiment)N/A
- LogS (predicted, ACD/Labs)(ph=7)-4.05
- LogSw (predicted, AB/LogsW2.0)0.01
- Sw (mg/ml) (predicted, ACD/Labs)0.07
- No.of HBond Donors4
- No.of HBond Acceptors14
- No.of Rotatable Bonds9
- TPSA188.9
- StatusFDA approved
- AdministrationN/A
- PharmacologyA cardiac glycoside. It is an acetyl derivative of digitoxin.
- Absorption_valueN/A
- Absorption (description)65
- Caco_2N/A
- Bioavailability70.0
- Protein binding80.0
- Volume of distribution (VD)N/A
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmN/A
- Half lifePlasma half-life, about 8 to 9 days.
- ExcretionIt is slowly excreted in the urine, about 20% of a dose being excreted in 6 days; digitoxin accounts for about 60% of the urinary material. About 15 to 20% of a dose is eliminated in the faeces over a period of 18 days.
- Urinary ExcretionN/A
- CleranceN/A
- ToxicityToxicity includes ventricular tachycardia or ventricular fibrillation, or progressive bradyarrhythmias, or heart block. LD50 = 7.8 mg/kg (orally in mice).
- LD50 (rat)N/A
- LD50 (mouse)N/A