- Molecular NamePosaconazole
- Synonymposaconazole
- Weight700.791
- Drugbank_IDDB01263
- ACS_NO171228-49-2
- Show 3D model
- LogP (experiment)N/A
- LogP (predicted, AB/LogP v2.0)5.39
- pkaN/A
- LogD (pH=7, predicted)5.38
- Solubility (experiment)N/A
- LogS (predicted, ACD/Labs)(ph=7)-4.73
- LogSw (predicted, AB/LogsW2.0)0.0
- Sw (mg/ml) (predicted, ACD/Labs)0.01
- No.of HBond Donors1
- No.of HBond Acceptors12
- No.of Rotatable Bonds12
- TPSA111.79
- StatusFDA approved
- AdministrationN/A
- PharmacologyA triazole antifungal drug.
- Absorption_valueN/A
- Absorption (description)N/A
- Caco_2N/A
- Bioavailability96.0
- Protein binding98.5
- Volume of distribution (VD)5~19 L/kg
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmN/A
- Half life16~31 h
- ExcretionFecal (77%) and renal (14%)
- Urinary ExcretionN/A
- CleranceN/A
- ToxicityN/A
- LD50 (rat)N/A
- LD50 (mouse)N/A