- Molecular NameRemikiren
- SynonymRo 42-5892
- Weight630.851
- Drugbank_IDDB00212
- ACS_NO126222-34-2
- Show 2D model
- LogP (experiment)2.75
- LogP (predicted, AB/LogP v2.0)2.77
- pkaN/A
- LogD (pH=7, predicted)2.4
- Solubility (experiment)N/A
- LogS (predicted, ACD/Labs)(ph=7)-5.5
- LogSw (predicted, AB/LogsW2.0)0.01
- Sw (mg/ml) (predicted, ACD/Labs)0.0
- No.of HBond Donors5
- No.of HBond Acceptors10
- No.of Rotatable Bonds16
- TPSA169.86
- StatusFDA approved
- AdministrationN/A
- PharmacologyA renin inhibitor under development for the treatment of hypertension (high blood pressure).
- Absorption_valueN/A
- Absorption (description)Absorbed following oral administration.
- Caco_2N/A
- Bioavailability1.0
- Protein binding83.0
- Volume of distribution (VD)70L
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmN/A
- Half lifeN/A
- ExcretionN/A
- Urinary ExcretionN/A
- CleranceN/A
- ToxicityN/A
- LD50 (rat)N/A
- LD50 (mouse)N/A