- Molecular NameLymecycline
- Synonym7-Chlorotetracycline; Chlorotetracycline; Chlorotetracycline hydrochloride; Chlortetracyclin; Chlortetracycline; Chlortetracycline hydrochloride; Chlortetracyclinium chloride; CLTC
- Weight602.641
- Drugbank_IDDB00256
- ACS_NO992-21-2
- Show 3D model
- LogP (experiment)-3.2
- LogP (predicted, AB/LogP v2.0)-3.03
- pkaN/A
- LogD (pH=7, predicted)-4.1
- Solubility (experiment)Soluble (at all physiological pH values)
- LogS (predicted, ACD/Labs)(ph=7)-2.07
- LogSw (predicted, AB/LogsW2.0)2.9
- Sw (mg/ml) (predicted, ACD/Labs)4.01
- No.of HBond Donors10
- No.of HBond Acceptors14
- No.of Rotatable Bonds10
- TPSA242.98
- StatusFDA approved
- AdministrationN/A
- PharmacologyA tetracycline broad-spectrum antibiotic
- Absorption_value100.0
- Absorption (description)Absorption is fast and efficient. Bioavailability is 100% following oral administration.
- Caco_2N/A
- Bioavailability100.0
- Protein bindingN/A
- Volume of distribution (VD)N/A
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmN/A
- Half lifeN/A
- ExcretionN/A
- Urinary ExcretionN/A
- CleranceN/A
- ToxicityAdverse effects include nausea, vomiting, diarrhoea, glossitis, enterocolitis, dysphagia, dermatitis, hypersensitivity reactions, proctitis, and vaginitis.
- LD50 (rat)N/A
- LD50 (mouse)N/A