- Molecular NameNetilmicin
- Synonym1-N-Ethylsisomicin
- Weight475.587
- Drugbank_IDDB00955
- ACS_NO56391-56-1
- Show 3D model
- LogP (experiment)-3.981
- LogP (predicted, AB/LogP v2.0)-5.26
- pkaN/A
- LogD (pH=7, predicted)-10.74
- Solubility (experiment)100 mg/ml
- LogS (predicted, ACD/Labs)(ph=7)0.32
- LogSw (predicted, AB/LogsW2.0)779.65
- Sw (mg/ml) (predicted, ACD/Labs)928.33
- No.of HBond Donors11
- No.of HBond Acceptors12
- No.of Rotatable Bonds8
- TPSA199.73
- StatusFDA approved; US withdrawn
- AdministrationInjection or infusion
- PharmacologyA member of the aminoglycoside family of antibiotics. These antibiotics have the ability to kill a wide variety of bacteria.
- Absorption_value0.0
- Absorption (description)Rapidly and completely absorbed after IM administration, peak serum levels were achieved within 30-60 minutes. Aminoglycosides are poorly absorbed from the gastrointestinal tract.
- Caco_2N/A
- Bioavailability0.0
- Protein binding10.0
- Volume of distribution (VD)N/A
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmNo evidence of metabolic transformation, typically 80% is recoverable in the urine within 24 hours
- Half life2.5 h
- ExcretionN/A
- Urinary ExcretionN/A
- CleranceN/A
- ToxicityNetilmicin has the potential to cause disturbances in balance and a hearing loss.
- LD50 (rat)N/A
- LD50 (mouse)N/A