- Molecular NameRemoxipride
- SynonymRemoxiprida [INN-Spanish]; Remoxipride [Usan:Ban:Inn]; Remoxipridum [INN-Latin]; Romoxipride
- Weight371.275
- Drugbank_IDDB00409
- ACS_NO117591-79-4
- Show 2D model
- LogP (experiment)2.13
- LogP (predicted, AB/LogP v2.0)2.62
- pka8.9
- LogD (pH=7, predicted)0.33
- Solubility (experiment)0.074 mg/ml
- LogS (predicted, ACD/Labs)(ph=7)-0.33
- LogSw (predicted, AB/LogsW2.0)0.17
- Sw (mg/ml) (predicted, ACD/Labs)1.24
- No.of HBond Donors1
- No.of HBond Acceptors5
- No.of Rotatable Bonds6
- TPSA50.8
- StatusFDA approved
- AdministrationN/A
- PharmacologyA psychoactive drug and substituted benzamide which was a promising antipsychotic during clinical trials in the 1990s, but was removed due to possible side effects.
- Absorption_value100.0
- Absorption (description)N/A
- Caco_2N/A
- Bioavailability90.0
- Protein binding80.0
- Volume of distribution (VD)0.5~0.7 L/kg
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmNo active metabolites
- Half life4~7 h
- ExcretionN/A
- Urinary ExcretionN/A
- CleranceN/A
- ToxicityN/A
- LD50 (rat)LD50=820 (intraperitoneal)
- LD50 (mouse)N/A