- Molecular NameRabeprazole
- SynonymIrsogladine Maleate; rabeprazole sodium; Rebeprazole sodium
- Weight359.45
- Drugbank_IDDB01129
- ACS_NO117976-89-3
- Show 3D model
- LogP (experiment)N/A
- LogP (predicted, AB/LogP v2.0)2.48
- pka5
- LogD (pH=7, predicted)2.47
- Solubility (experiment)N/A
- LogS (predicted, ACD/Labs)(ph=7)-3.74
- LogSw (predicted, AB/LogsW2.0)0.32
- Sw (mg/ml) (predicted, ACD/Labs)0.06
- No.of HBond Donors1
- No.of HBond Acceptors6
- No.of Rotatable Bonds8
- TPSA96.31
- StatusFDA approved
- AdministrationN/A
- PharmacologyAn antiulcer drug in the class of proton pump inhibitors.
- Absorption_value90.0
- Absorption (description)N/A
- Caco_2N/A
- Bioavailability52.0
- Protein binding96.3
- Volume of distribution (VD)N/A
- Blood/Plasma Partitioning ratio (D_blood)N/A
- MetabollsmMostly non-enzymatic, partly hepatic (CYP2C19)
- Half life1~2 h
- Excretion90% renal
- Urinary ExcretionN/A
- CleranceN/A
- ToxicityThe most common side effects of Rabeprazole are diarrhea, nausea, vomiting, constipation, rash and headaches. Dizziness, nervousness, abnormal heartbeat, muscle pain, weakness, leg cramps and water retention rarely occur.
- LD50 (rat)N/A
- LD50 (mouse)N/A