6BV8

Target information

RCSB PDB
6BV8
Title
Structure of proteinaceous RNase P 1 (PRORP1) from A. thaliana complexed with Mn after 3-hour soak with juglone
Method
X-RAY DIFFRACTION
Resolution
2.1
Classification
HYDROLASE/HYDROLASE INHIBITOR
Organism
Arabidopsis thaliana
Protein
Proteinaceous RNase P 1, chloroplastic/mitochondrial (Q66GI4)
Year
2017
Publication Title
Inhibition of protein-only RNase P with Gambogic acid and Juglone
Abstract

Not Available

External Link
RCSB PDB





Ligand information

HET
JUG
Chain ID
A
HET Number
601
Molecular Formula
C10H6O3
Structure
2D structure
IUPAC Name
5-hydroxynaphthalene-1,4-dione
InChI
InChI=1S/C10H6O3/c11-7-4-5-9(13)10-6(7)2-1-3-8(10)12/h1-5,12H
InChI Key
KQPYUDDGWXQXHS-UHFFFAOYSA-N
Canonical SMILES
Oc1cccc(c12)C(=O)C=CC2=O
Bioactivity data
CI000005

Covalent Binding

Warhead
Michael Acceptor
Reaction Mechanism
Michael Addition
Residue
CYS : 353
Residue Chain
A
Interactions
Pharmacophore Model